Small molecules used in screening
17-AAG | CHIR258 | JAK1i | Nilotinib | SB-43152 |
8 Azaguanine | CHIR265 | JAK3i | P38i | SB203580 |
ABT-864 | CI-1033 | JNK2i | Pan-JAKi | Sorafenib |
Adiphenine | CP-690550 | JNKIIi | PD153035 | SRCi |
AG490 | CYC-202 | KN92 | PD325901 | Staurosporine |
AKTIV | Dasatinib | KN93 | PD98059 | STO609 |
AKTX | EGFRi | Lapatinib | PI-103 | Sunitinib |
AMPK | Erlotinib | LSD1 | Piperine | SYKi |
Anisomycin | Estradiol | LY294002 | PKC412 | Thapsigargin |
AZD-1152 | Gefitinib | LY333531 | PP2 | Trichostatin A |
Azithromycin | Go6976 | MEK1/2 | Proguanil | Tunicamycin |
BAY-11 | GW-786034 | Menadione | PTK787 | Vorinostat |
BIRB-796 | H-89 | MLN-8054 | R1881 | VX-680 |
Boldine | Harmane | MLN518 | Resveratrol | Zardaverine |
cAMP | Imatinib | QNZ | SB-202190 | ZD-6474 |
17-AAG | CHIR258 | JAK1i | Nilotinib | SB-43152 |
8 Azaguanine | CHIR265 | JAK3i | P38i | SB203580 |
ABT-864 | CI-1033 | JNK2i | Pan-JAKi | Sorafenib |
Adiphenine | CP-690550 | JNKIIi | PD153035 | SRCi |
AG490 | CYC-202 | KN92 | PD325901 | Staurosporine |
AKTIV | Dasatinib | KN93 | PD98059 | STO609 |
AKTX | EGFRi | Lapatinib | PI-103 | Sunitinib |
AMPK | Erlotinib | LSD1 | Piperine | SYKi |
Anisomycin | Estradiol | LY294002 | PKC412 | Thapsigargin |
AZD-1152 | Gefitinib | LY333531 | PP2 | Trichostatin A |
Azithromycin | Go6976 | MEK1/2 | Proguanil | Tunicamycin |
BAY-11 | GW-786034 | Menadione | PTK787 | Vorinostat |
BIRB-796 | H-89 | MLN-8054 | R1881 | VX-680 |
Boldine | Harmane | MLN518 | Resveratrol | Zardaverine |
cAMP | Imatinib | QNZ | SB-202190 | ZD-6474 |
For each molecule, at least 3 doses were tested. Cell viability was quantified using the 3-(4,5-dimethylthiazol-2-yl)-5-(3-carboxymethoxyphenyl)-2-(4-sulfophenyl)-2H-tetrazolium assay.