Table 2.

Specific GR binding sites/cell (Bmax) and receptor affinity for ligand (KD) values for ALL xenografts


Xenograft

Bmax (sites/cell)

KD (nM)
ALL-2   9 762 ± 446   8.4 ± 1.3  
ALL-3   8 931 ± 314   5.9 ± 0.7  
ALL-4   6 555 ± 222   4.6 ± 0.6  
ALL-7   15 794 ± 543   4.1 ± 0.6  
ALL-8   1 752 ± 140   5.5 ± 1.6  
ALL-10   8 713 ± 435   11.0 ± 1.8  
ALL-16   7 117 ± 247   4.9 ± 0.7  
ALL-17   8 772 ± 236   3.9 ± 0.5  
ALL-18   9 432 ± 296   5.3 ± 0.6  
ALL-19
 
7 149 ± 294
 
2.7 ± 0.5
 

Xenograft

Bmax (sites/cell)

KD (nM)
ALL-2   9 762 ± 446   8.4 ± 1.3  
ALL-3   8 931 ± 314   5.9 ± 0.7  
ALL-4   6 555 ± 222   4.6 ± 0.6  
ALL-7   15 794 ± 543   4.1 ± 0.6  
ALL-8   1 752 ± 140   5.5 ± 1.6  
ALL-10   8 713 ± 435   11.0 ± 1.8  
ALL-16   7 117 ± 247   4.9 ± 0.7  
ALL-17   8 772 ± 236   3.9 ± 0.5  
ALL-18   9 432 ± 296   5.3 ± 0.6  
ALL-19
 
7 149 ± 294
 
2.7 ± 0.5
 
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