Table 1.
Kinase profiles of current JAK2 inhibitors
Kinase
.
Enzyme IC
50
, nM
.
Fedratinib
.
Ruxolitinib
.
Pacritinib
.
Momelotinib
.
JAK1
105
3.3
1280
11
JAK2
3
2.8
23
18
JAK3
1002
428
520
155
TYK2
405
19
50
17
Kinase
.
Enzyme IC
50
, nM
.
Fedratinib
.
Ruxolitinib
.
Pacritinib
.
Momelotinib
.
JAK1
105
3.3
1280
11
JAK2
3
2.8
23
18
JAK3
1002
428
520
155
TYK2
405
19
50
17
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