The saliva of hemovores, such as ticks, contains many anticoagulant molecules, which prevent the host from clotting so that the hemovore may feed. De Paula et al demonstrated that 1 tick anticoagulant, Ixolaris, works by binding the TF/FVIIa/FXa complex, similar to human TFPI. However, unlike TFPI, Ixolaris binds an exosite on FXa that induces a conformational change in its active site and loss of proteolytic function, a newly uncovered mechanism for regulating FXa function and limiting coagulation.

The saliva of hemovores, such as ticks, contains many anticoagulant molecules, which prevent the host from clotting so that the hemovore may feed. De Paula et al demonstrated that 1 tick anticoagulant, Ixolaris, works by binding the TF/FVIIa/FXa complex, similar to human TFPI. However, unlike TFPI, Ixolaris binds an exosite on FXa that induces a conformational change in its active site and loss of proteolytic function, a newly uncovered mechanism for regulating FXa function and limiting coagulation.

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